http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2018502925-A

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filingDate 2016-01-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2018-02-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2018502925-A
titleOfInvention Compounds and methods for targeted androgen receptor degradation
abstract The present invention relates to bifunctional compounds that are useful for degrading (and inhibiting) androgen receptors. In particular, the present invention includes at one end a VHL ligand that binds to a ubiquitin ligase such that the androgen receptor is placed in close proximity to the ubiquitin ligase to effect degradation (and inhibition) of the androgen receptor, The present invention relates to a compound comprising a moiety that binds to the body at the other end. The present invention exhibits a wide range of pharmacological activities associated with the compounds of the present invention, consistent with androgen receptor degradation / inhibition.
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID564123
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1LZI1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ27404
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP62976
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB3NWW9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP19114
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP04707
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP62972
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID163800002
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP21898
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5HRD6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO62641
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ66KB0
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID326237
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ07295
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8MXJ7
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID482154
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID25610
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID6573232
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID3873815
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0CS17
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID334380
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID466449529
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP54855
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24335
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP08157
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0CS16
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP48815
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6CUD9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP48814
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP48977
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ63886
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ28746
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5PJC4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9HAW8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA6ZTT5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9C9Y7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO02837
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9C918
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID467151
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP05016
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP21300
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP13603
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9C8X7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP06525
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ80X89
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID443
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6DG60
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP41751
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO02663
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID101256912
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP12886
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6FQK7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP12854
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5PKP9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP21518
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9XT55
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP97712
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP61086
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP25867
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP15121
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID828049
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP25866
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID102144258
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO74187
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100002479
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP25865
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID6567587
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8BWQ1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4H9W2
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID886306
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO60218
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ64133
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6UWM9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP80360
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP00328
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ06AA9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA8WLF6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP48617
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP22589
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP00327
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP00326
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9JJZ4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP25869
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP80338
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4MA02
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP25868
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP80467
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4L7V4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ96XE0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP27949
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4JKB7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ28513
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ47898
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP22570
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID3355109
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID3919406
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO07737
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4IF39
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6C093
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP19854
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0A5C1REZ4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8L7T3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP19848
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6BYG4
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID490325
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4R6G1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6BU36
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP48750
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4Q2J2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP48749
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP78717
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6ZQM8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4N208

Total number of triples: 1081.