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filingDate 2015-11-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2018-02-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2018502901-A
titleOfInvention Methods for producing prodrugs and targeted therapeutic compounds
abstract A method for preparing the compound of Formula 1 is provided. Various compounds utilized in the method are also provided, wherein a method of preparing these compounds provided XO-CO- (CH 2) n NH 2. Also provided is a compound having (where n is an integer greater than 2). Further provided is a method of making the compound. Further provided is a method of producing a prodrug of a biologically active compound. [Selection] Figure 1
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