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publicationDate 2018-02-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2018502851-A
titleOfInvention Simple synthesis of urea derivatives of amphotericin B
abstract Certain derivatives of amphotericin B (AmB) are provided that are characterized by reduced toxicity and retention of antifungal activity. Some of the derivatives are AmB C16 urea derivatives and C16 carbamate derivatives. A method for producing an AmB derivative is also disclosed.
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