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inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_192ef7f36cd7bd5c37b5f650069d4b03
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publicationDate 2018-05-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2018083816-A
titleOfInvention Novel conjugates comprising TETRA GALNAC and peptides and methods for delivering oligonucleotides
abstract The present invention provides a new single chemical conjugate capable of effectively performing delivery efficiency, cellular uptake and / or endosome escape. 1) oligonucleotide; 2) one or more tetraGalNAc ligands of formula (I); optionally 3) one or more linkers; 4) one or more having a specific sequence And optionally 5) a modular composition comprising one or more targeting ligands, solubilizers, pharmacokinetic agents, lipids and / or masking agents. [Selection figure] None
priorityDate 2012-05-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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