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assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_bb75b0b19820e3833ebdcb31603b242b
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P43-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-4245
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D271-06
filingDate 2017-10-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1216428faef4d608c78af1bbf4a99dc4
publicationDate 2018-05-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2018070607-A
titleOfInvention Method for producing oxadiazole derivative substituted with amino group
abstract An intermediate of an oxadiazole derivative substituted with an amino group and having an NPY Y5 receptor antagonistic activity, and a production method thereof. The compound represented by formula (I) is selected from substituted / unsubstituted imidazole, substituted triazole, substituted pyrazole, substituted pyrrole, substituted / unsubstituted benzimidazole, substituted benzotriazole, and substituted benzopyrazole. An intermediate that is a salt with one basic compound. Oxadi substituted with an amino group having NPY Y5 receptor antagonistic activity comprising reacting the salt with a halogenating agent and a base, optionally in the presence of a basic compound forming the salt A method for producing an azole derivative. [Selection figure] None
priorityDate 2016-10-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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