http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2017516817-A

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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P23-00
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P25-04
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filingDate 2015-06-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2017-06-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2017516817-A
titleOfInvention Amide derivatives of 1-oxa-4,9-diazaspiroundecane compounds having various activities against pain
abstract The present invention relates to compounds having dual pharmacological activity for both sigma (σ) receptors and μ-opioid receptors, more specifically diazaspiroundecane compounds having this pharmacological activity, It relates to a process for the preparation of such compounds, pharmaceutical compositions containing them and their use in therapy, in particular for the treatment of pain. [Chemical 1] Where Y is [Chemical formula 2] And n is 1 or 2; q is 1, 2, 3, 4, 5 or 6; X is a bond, —C (O) O—, —C (O) NR 8 —, —C (O) —, —O— or —C (R 4 R 4 ′ ) —; R 1 is C (O) R 5 or S (O) 2 R 5 .
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2017535566-A
priorityDate 2014-06-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID414701355
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID451273111
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID304271
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID414392184
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118562298
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID798
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419559546
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12732
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7369
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428932000
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID411322314
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID18373917
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID447941571
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID8082
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11185
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428932076
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4837
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121306019
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118562191
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419521555
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5344
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID130202753
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458394722
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419488216
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421297261
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Total number of triples: 388.