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filingDate 2017-03-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_65489a6ac67f9e41137c3b91345b424c
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b43b747bb98b02fac11bce5e5c494360
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publicationDate 2017-10-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2017178941-A
titleOfInvention Composition for inhibiting androgen-dependent or independent prostate cancer cells and pharmaceutical preparation for prostate cancer containing the same
abstract [PROBLEMS] To suppress the activation of androgen receptor, which is used for prostate cancer, is effective in suppressing androgen-dependent or independent growth of prostate cancer, and has an effect even if AR-V7 is expressed. Provided are a composition for suppressing androgen-dependent or independent prostate cancer cells that is effective against an anticancer drug-resistant cell line, and a pharmaceutical preparation for prostate cancer using the same. A composition for inhibiting androgen-dependent or independent prostate cancer cells has the chemical formula (1) [Chemical 1] (X- is a hydrocarbon aromatic ring group or aromatic heterocyclic group, Y 1 -and Y 2 -are both or one is a hydrocarbon aromatic ring group or aromatic heterocyclic group, the other is a hydrogen atom, Z = is a bonded carbon Α, β-saturated or unsaturated represented by an atom or a functional group that forms or forms a ketone group, a thioketone group, an imino group, or an oxime group with an atom, and Y 3 -represents a hydrogen atom, a perhalogeno hydrocarbon group, etc. Including a ketone derivative or a pharmaceutically acceptable salt thereof. A pharmaceutical preparation for prostate cancer contains this composition. [Selection figure] None
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