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publicationDate 2017-04-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2017070299-A
titleOfInvention Modification of antisense compounds
abstract An antisense oligonucleotide with improved binding affinity and nuclease resistance is provided. An antisense oligonucleotide comprising at least one modification incorporated between two bases of an antisense oligonucleotide, the modification increasing the binding affinity and nuclease resistance of the antisense oligonucleotide, An antisense oligonucleotide comprising at least one modification within three nucleotide bases, wherein the modification is a naphthylene-azo compound represented by the following formula: [Selection figure] None
priorityDate 2010-09-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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