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filingDate 2014-11-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2016-11-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2016535097-A
titleOfInvention 4- (Indol-3-yl) -pyrazole derivatives, pharmaceutical compositions and methods for use
abstract The present invention relates to a compound of formula (I), or a pharmaceutically acceptable enantiomer, salt or solvate thereof. The invention further relates to the use of compounds of formula I as tryptophan 2,3-dioxygenase (TDO2) inhibitors. The present invention relates to the use of compounds of formula I for the treatment and / or prevention of cancer, Parkinson's disease, neurodegenerative disorders such as Alzheimer's disease and Huntington's disease, chronic viral infections such as HCV and HIV, depression and obesity Also related. The invention also relates to a process for preparing the compound of formula (I). [Chemical 1]
priorityDate 2013-11-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118060232
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP49319
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID109644000
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP49318
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID315017
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID351278
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID19354
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID15655
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID76980
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118060436
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122513730
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ27710
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP49315
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7369
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7915
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415914699
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP49284
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450461534
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID422483787
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ27487
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419571630

Total number of triples: 956.