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filingDate 2014-06-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2016-09-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2016528179-A
titleOfInvention Production method and crystal form of MDM2 inhibitor
abstract The present invention relates to 2-((3R, 5R, 6S) -5- (3-chlorophenyl) -6- (4-chlorophenyl) -1-((S) -1- (isopropylsulfonyl) -3-methylbutane-2. A method for producing -yl) -3-methyl-2-oxopiperidin-3-yl) acetic acid and intermediates, and a method for producing intermediates are provided. Also provided are crystalline forms of the compounds and intermediates.
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