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filingDate 2014-07-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2016-08-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2016523941-A
titleOfInvention Modified BET protein inhibitory dihydroquinoxalinones and dihydropyridopyrazinones
abstract The present invention relates to general formula (I) BET protein inhibition, particularly BRD4 inhibition, wherein A, X, R 1 , R 2 , R 3 , R 4 , R 5 , R 6 and n are each as defined in the specification Dihydroquinoxalinones and dihydropyridopyrazinones, intermediates for the preparation of the compounds of the invention, pharmaceutical compositions comprising the compounds of the invention, and in cases of hyperproliferative disorders, in particular neoplastic disorders Relating to its prophylactic and therapeutic use. The invention further relates to the use of BET protein inhibitors in viral infections, neurodegenerative disorders, inflammatory diseases, atheropathic disorders and male fertility control. [Chemical 1]
priorityDate 2013-07-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID432778507
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP05004
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6336229
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID432778515
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP05012
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5394
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ28819
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID432778554
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450737290
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID432778115
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID87056098
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2733084
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID18033
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3015207
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID412782985
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID424497431
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID117800713
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121412238
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO62641
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID432777613
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID432778391
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID87056100
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ90YI0
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID121412240
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450024818
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID179337
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID432777660
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID25080282
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID78688
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID432777706
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID432777455
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11167602
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419486648
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID455824109
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID432777874
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID87055453
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID416010490
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419501829
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID432777062
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID448118596
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0A3Q1MKE9
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID432777397
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Total number of triples: 1337.