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filingDate 2013-12-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2016-04-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2016512240-A
titleOfInvention Fluorescence imaging of inflammatory diseases with ligands conjugated with fluorescent compounds
abstract The present disclosure relates to compounds useful as near-infrared fluorescent probes, comprising i) a pteroyl ligand that binds to a target receptor protein, ii) a dye molecule, and iii) a linker molecule comprising an amino acid or derivative thereof. . The present disclosure further describes a method for imaging inflammatory diseases using the compounds. The present disclosure provides a method for treating inflammatory diseases by using an effective amount of an amino acid linking group conjugated with a compound used for targeted imaging of inflamed tissue and lymph nodes.
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