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filingDate 2014-03-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2016-04-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2016510772-A
titleOfInvention Tetracyclic bromodomain inhibitors
abstract The present invention relates to compounds of formula (I) that are useful as agents in the treatment of diseases and conditions including inflammatory diseases, cancer and AIDS wherein R 1 , R 2 , R 6 , Y 1 , Y 2 , Y 3 , A 1 , A 2 , A 3 and A 4 have any of the values defined herein. And pharmaceutically acceptable salts thereof. Also provided are pharmaceutical compositions comprising one or more compounds of formula (I).
priorityDate 2013-03-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID12043
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCD4A9I5
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419502640
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID431778410
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7401
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCD4A1A6
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID140890567
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID458294
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5381
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135413520
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO77812
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCD3ZQL7
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428988562
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5379
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419551313
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP54107
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID414866614
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID89656147
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421256454
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428988522
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID431904250
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID1989
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7YRB5
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID416154167
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID3002
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID314856
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID118465075
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID378478
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID140890512
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID392622
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Total number of triples: 2908.