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filingDate 2013-12-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2016-02-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2016503805-A
titleOfInvention Substituted pyrimidine aminoalkyl-quinazolones as phosphatidylinositol 3-kinase inhibitors
abstract The disclosure provides a phosphatidylinositol 3-kinase (PI3K) inhibitor of formula (I), or a pharmaceutically acceptable salt thereof, wherein R 1 , R 2 , n, R 3 , R 4 , R 5 and R 6 are as defined herein. These compounds are useful for the treatment of conditions mediated by one or more PI3K isoforms, such as PI3Kδ. The present disclosure further provides pharmaceutical compositions comprising a compound of formula (I) or a pharmaceutically acceptable salt thereof, as well as to treat a condition mediated by one or more PI3K isoforms such as PI3Kδ. Methods of using these compounds and compositions are provided.
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID90233050
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID448151510
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ92087
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID90232783
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP70091
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11273
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID31722
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419503366
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP20809
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419576231
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID445580
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ92112
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP20808
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426391582
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID39562
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ92111
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP58022
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID90233179
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID445643
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3005573
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID360918
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID90233045
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID90232800
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID417776695
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP30919
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID76286380
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID90233024
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID22341
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457502397
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID41210
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID439693
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419545072
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID76286379
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID281408
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID90233023
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457501988
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP40226
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID6612803
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID408869260
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID90233026
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3011155
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419545322
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393705
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID90232794
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID18343
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID535622
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP30918

Total number of triples: 1299.