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publicationDate 2016-01-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2016501374-A
titleOfInvention Compositions and methods for determination of FKBP-binding immunosuppressive drugs
abstract Disclosed is a composition for releasing an FKBP-bound immunosuppressive drug from an endogenous binding substance in a sample suspected of containing the FKBP-bound immunosuppressive drug. The composition comprises a sirolimus derivative modified with a bulky organic group at the triene portion of the sirolimus molecule. The composition may be used in conjunction with assays for FKBP-binding immunosuppressive drugs in samples suspected of containing FKBP-binding immunosuppressive drugs.
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