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filingDate 2015-04-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c95651d1f7ed0ae5021d75308336826f
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publicationDate 2015-08-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2015155430-A
titleOfInvention Synthetic macrocyclic compounds with fixed conformation
abstract The present invention provides a novel macrocyclic compound exhibiting agonistic or antagonistic activity against a motilin receptor, a serotonin receptor and a prostaglandin F2A receptor. A macrocyclic compound represented by formula (I) in which building blocks A, B and C are incorporated. [Efficacy] It is effective for the treatment of hypokinetic disorders of the gastrointestinal tract, CNS related diseases and ocular hypertension. [Selection figure] None
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