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filingDate 2012-09-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2014-10-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2014527997-A
titleOfInvention 5-Benzylaminomethyl-6-aminopyrazolo [3,4-B] pyridine derivatives as cholesteryl ester transfer protein (CETP) inhibitors useful for the treatment of atherosclerosis
abstract This application relates to a series of substituted pyrazolopyridin-6-amines having the general formula (I), including their stereoisomers and / or their pharmaceutically acceptable salts. In which R, R 1 , R 2 , R a , R aa , R b and n are as defined herein. The invention further relates to pharmaceutical compositions comprising a compound of formula (I). The compounds of the present application are useful as CETP inhibitors for increasing HDL cholesterol and decreasing LDL cholesterol in patients.
priorityDate 2011-09-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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