http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2014509640-A

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http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-06
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http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D307-80
classificationIPCAdditional http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-343
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D307-80
filingDate 2012-03-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2014-04-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2014509640-A
titleOfInvention Process for the preparation of dronedarone by N-butylation
abstract The present invention relates to a novel process for preparing dronedarone (I) and pharmaceutically acceptable salts thereof, wherein the compound of formula (II) or a salt thereof is represented by the formula L— (CH 2 ) 3 —CH 3 (III) Reaction with a compound of formula (wherein L is a leaving group), the resulting product is isolated and optionally converted to its pharmaceutically acceptable salt. The invention also relates to some novel intermediate compounds and their preparation.
priorityDate 2011-03-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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