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filingDate 2011-11-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2013-12-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2013544811-A
titleOfInvention Heterocyclic compounds as S1P1 agonists for the treatment of autoimmune and vascular diseases
abstract Compound of formula (I) Or a stereoisomer, salt or prodrug thereof, wherein W is CH 2 or O; And R 1 , R 2 , R 3 , R 4 , n and G are as described herein, a compound or a stereoisomer, salt or prodrug thereof is disclosed. Also disclosed are methods of using such compounds as selective agonists for the G protein coupled receptor S1P 1 and pharmaceutical compositions comprising such compounds. These compounds are useful in the treatment, prevention or delay of progression of diseases or disorders in various medical fields such as autoimmune diseases and vascular diseases.
priorityDate 2010-11-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 488.