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filingDate 2011-09-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2013-10-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2013538235-A
titleOfInvention Macrocyclic proline-derived HCV serine protease inhibitor
abstract The present invention discloses compounds of formula (I) or pharmaceutically acceptable salts, esters or prodrugs thereof which inhibit serine protease activity, in particular hepatitis C virus (HCV) NS3-NS4A protease activity. Formula (I) is disclosed. Therefore, the compound of the present invention interferes with the life cycle of hepatitis C virus and is still useful as an antiviral agent. The present invention further relates to pharmaceutical compositions comprising the aforementioned compounds for administration to a subject suffering from HCV infection. The invention also relates to a method for treating HCV infection in a subject by administering a pharmaceutical composition comprising a compound of the invention.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2021113192-A
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2017509670-A
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