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filingDate 2011-04-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2013-06-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2013525417-A
titleOfInvention Sustained release pharmaceutical composition of brivaracetam
abstract The present invention relates to a sustained release pharmaceutical composition comprising brivaracetam or a pharmaceutically acceptable derivative thereof. Further disclosed is a sustained release pharmaceutical composition comprising a core and a coating agent surrounding the core, wherein the core includes brivaracetam or a pharmaceutically acceptable derivative thereof, A hydrophobic release control agent is included. The sustained release pharmaceutical composition includes brivaracetam or a pharmaceutically acceptable derivative thereof and a hydrophobic release control agent, wherein the composition is a USP apparatus in 900 ml of pH 6 phosphate buffer solution. At least 80% brivaracetam elutes between about 7 and about 24 hours as measured using type II at 50 rpm and 37 ° C. Also disclosed is a sustained release pharmaceutical composition useful for the treatment of epilepsy and symptomatic myoclonus comprising brivaracetam or a pharmaceutically acceptable derivative thereof and a hydrophobic release controlling agent.
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type http://data.epo.org/linked-data/def/patent/Publication

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