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filingDate 2010-11-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2013-03-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2013510870-A
titleOfInvention Spiropiperidine compounds as ORL-1 receptor antagonists
abstract An ORL-1 receptor antagonist of the formula: , Its use, and its method of preparation. ORL-1 antagonists are considered useful for the treatment of depression and / or for the treatment of overweight, obesity, and / or weight maintenance after treatment of overweight or obesity. Certain compounds have also been demonstrated by animal models that the compounds of the present invention are useful for the treatment of migraine.
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Total number of triples: 505.