abstract |
Disclosed are GABA B receptor ligands γ-aminobutyric acid derivatives of formula (I), pharmaceutical compositions containing such derivatives, and methods of using such derivatives and pharmaceutical compositions thereof to treat diseases. R 5 is selected from —COOH, —SOOH, and —P (O) (OH) R 8 , wherein R 8 is selected from hydrogen and C 1-4 alkyl. [Selection figure] None |