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filingDate 2010-03-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2012-09-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2012520859-A
titleOfInvention SHP90 inhibitory indazole derivatives, compositions containing them, and uses thereof
abstract The present invention relates to novel products having the formula (I), wherein R4 represents H, CH3, CH2CH3, CF3, F, Cl, Br, I; Het is one or more R1 or R′1 Represents a heterocycle optionally substituted by a group, wherein the one or more R1 or R'1 groups are H, halogen, CF3, nitro, cyano, alkyl, hydroxy, mercapto, amino, alkylamino, dialkylamino, Alkoxy, phenylalkoxy, alkylthio, carboxy, carboxamide, CO-NH (alkyl), CON (alkyl) 2, NH-CO-alkyl, sulfonamide, NH, free or esterified with an alkyl group Selected from -SO2-alkyl, S (O) 2-NHalkyl, S (O2) -N (alkyl) 2, All of the alkyl, alkoxy and alkylthio groups are optionally substituted; R is selected from the group comprising (A ′), (B), (C), (D) and (E), wherein W1, W2 and W3 independently represent CH or N, X represents O, S, NR2, C (O), S (O) or S (O) 2, and V represents H, Hal, —O—R 2 or —NH—R 2, where R 2 represents H, optionally substituted alkyl, cycloalkyl or heterocycloalkyl. It relates to products which are in isomeric form and their salts and are intended for use as drugs.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2016511237-A
priorityDate 2009-03-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 921.