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filingDate 2009-08-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2012-01-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2012500794-A
titleOfInvention [4- (5-Aminomethyl-2-fluoro-phenyl) -piperidin-1-yl]-[7-fluoro-1- (2-methoxy-ethyl) -4-trifluoromethoxy- as mast cell tryptase inhibitor 1H-Indol-3-yl] -methanone
abstract The present invention relates to indole benzylamine compounds useful as tryptase inhibitors. Furthermore, the invention relates to the use of a compound for treating a patient suffering from or susceptible to a physiological condition in need of improvement by inhibition of tryptase, comprising administering to the patient a therapeutically effective amount of the compound. To do. The present invention further relates to pharmaceutical compositions comprising a therapeutically effective amount of a compound of formula I and a pharmaceutically acceptable carrier. [Chemical 1]
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2013502425-A
priorityDate 2008-08-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 428.