http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2012105640-A

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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/G01N33-50
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filingDate 2011-10-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_2fcfbcc56fa8f84a3e72d96c9e85bf42
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publicationDate 2012-06-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2012105640-A
titleOfInvention Method for screening drug candidate compound for Gs-coupled receptor
abstract Provided is a method for screening a drug candidate compound for a Gs-coupled receptor that activates the Gs-coupled receptor and does not cause desensitization. It has been found that by using a partial agonist activity for a Gs-coupled receptor as an index, a compound that activates the Gs-coupled receptor and does not cause desensitization can be efficiently screened. At least one receptor selected from the group consisting of a β1 adrenergic receptor, a β2 adrenergic receptor, a β3 adrenergic receptor, and a GLP-1 receptor. [Selection figure] None
priorityDate 2010-10-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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