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filingDate 2009-01-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2011-04-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2011511002-A
titleOfInvention Intralymphatic chemotherapy drug carrier
abstract A chemotherapeutic composition for subcutaneous administration can be constructed that is due to preferential lymphatic accumulation but also provides a therapeutic systemic concentration that is not toxic. The composition may comprise a pharmaceutically acceptable carrier and a nanoconjugate configured for preferential lymphatic accumulation after subcutaneous administration. The nanoconjugate may comprise a nanocarrier configured for preferential lymphatic accumulation after subcutaneous or intrastitial administration and a plurality of chemotherapeutic agents coupled to the nanocarrier. The nanoconjugate may have a dimension of about 10 to about 50 nm. The nanoconjugate may also be loaded with about 10 to about 50% w / w chemotherapeutic agent. The nanocarrier may be a hyaluronic acid polymer of about 3 kDa to about 50 kDa. Alternatively, the nanocarrier may be a dendrimer. [Selection] Figure 1 (A)
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