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filingDate 2008-10-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2011-01-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2011500727-A
titleOfInvention Bicyclic heterocyclic derivatives and their use as modulators of GPR119 activity
abstract The invention relates to bicyclic heterocycle derivatives, compositions comprising bicyclic heterocycle derivatives, and to treat or prevent obesity, diabetes, metabolic disorders, cardiovascular diseases or GPR119 activity related disorders in patients. The present invention relates to a method using a cyclic heterocyclic derivative. Compounds of formula (I), (II), (III) and (IV) and their pharmaceutically acceptable salts, solvates, esters or prodrugs (herein referred to as “bicyclic heterocyclic derivatives”) Can be useful for treating or preventing obesity, diabetes, diabetic complications, metabolic syndrome, cardiovascular disease or GPR119 activity-related disorders (each of which is a “medical condition”) in a patient. .
priorityDate 2007-10-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9A8T2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WKA2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9AAR7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68989
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68988
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB3QS41
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9NBU5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68987
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB1IGD3
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ4UMQ8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0ALU7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9GTW9
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID7939554
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5M2D4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7GXT4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3A6M6
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5360545
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9GTW8
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID467673418
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID291437
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP48097
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3ZZQ3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB3QNN0
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID420225124
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID182236
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5360515
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5FZU4
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID396488
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID7017737
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WKC5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ57CS9
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID163637190
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WKC4
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID8070
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11155794
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID416145391
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA7NBG3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA3CT21
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WKC3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9R0Q7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO73727
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID32
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA1KJU9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WKC2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCD4A9L7
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6992810
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WKC1
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID3921488
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WKC0
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID7017083
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP69441
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419536312
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WKB9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2HCV5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP69439
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WKB8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4TMG6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WKB7
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID57569763
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419508829
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID61614909
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA1KGL4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WKB6
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID107378852
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID414671823
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WKB5
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID147616393
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8PKU2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WKB4
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID888567
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2GJ13
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID56144
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12956
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB0T0C5
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419491887
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WKB3
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID853086
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID119440
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID404209
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID441314
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WKB2
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3961
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2735739
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID325875
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66173
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2NV57
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419551193
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID14496
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0QB12
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA3D5M6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WKB1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP69102
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0Q812
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0C0R4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP69101
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0C0R3
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID6803421
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11323257
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID521305
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP69048
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415733454
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426285296
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0B9A2
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID245822
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID23676156
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP69047
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3Z4S5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA1KT73
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID76218
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP69046
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID58270311
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8P8U7
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID424486649
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415140199
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP69045
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419579328
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB8D813
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421089475
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5FMV7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ706D1
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419492227
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1472986
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA1KQD8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ706D0
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID29230
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID26873
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419503925

Total number of triples: 2352.