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filingDate 2011-06-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_ac2211345ecd32464b3af910514bfed2
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_fea17fb9684ee5513d95d18167b96d0b
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publicationDate 2011-10-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2011213727-A
titleOfInvention Prodrugs of hyperbranched polymers
abstract A water-soluble prodrug is provided. The prodrug of the present invention comprises a water-soluble polymer having three or more branches, at least three of which are covalently bound to an active substance (eg, a small molecule). The composite of the present invention provides an optimal balance of polymer size and structure to achieve improved drug loading, which is the release of the complex of the present invention over a multi-branched water soluble polymer. This is because it has three or more active substances that can be combined. The prodrugs of the present invention are therapeutically effective and exhibit improved properties in vivo when compared to the unmodified parent drug. [Selection figure] None
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/KR-20150103749-A
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2014532714-A
priorityDate 2003-09-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24241
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419510530
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419535942
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415791472
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6AXU0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP20392
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID368436
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419506927
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WGZ9
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2202
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID650
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID463288
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID403657
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID617960
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID744785
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9XT83
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP80298
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ44056
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9XT84
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP20391
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID408035
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCH0ZG98
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66628747
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID454973655
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID467655129
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419503719
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ62935
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID744975
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP10145
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6V919
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID20604
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID467655170
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419503618
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419493889
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID403795
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419593172
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419504915
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419590905
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP35393
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415732864
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP20607
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCH0ZNW5
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9815560
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP48248
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP35391
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID454364416
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP70160
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4086
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5773
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID408786858
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP10424
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO00300
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID469423
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135515469
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458392451
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID25317
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5942
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1HFN3
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID408799882
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5780
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419591639
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9XS58

Total number of triples: 1354.