Predicate |
Object |
assignee |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_d12b0f56aeb4c6c528c7d3ca3573cdb7 |
classificationCPCAdditional |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07B2200-07 |
classificationCPCInventive |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C219-30 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C227-34 |
classificationIPCAdditional |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07B57-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07B61-00 |
classificationIPCInventive |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C213-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C229-34 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C219-28 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C227-16 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C227-34 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C215-54 |
filingDate |
2010-10-28-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
inventor |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8478908f0700473fd7024590afc0adec http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_40b949f3b107873cd4dad06472ce9dd2 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c41acf4f173bf2666660ad7f3fb7f346 |
publicationDate |
2011-05-26-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber |
JP-2011102295-A |
titleOfInvention |
Process for producing fesoterodine |
abstract |
From low cost starting materials of isobutyric acid (R) -2- (3-diisopropylamino-1-phenylpropyl) -4- (hydroxymethyl) phenol (fesoterodine) and its (S) enantiomer, high Providing an efficient synthesis method that is pure and can be reproduced on an industrial scale. A racemic compound of formula II is resolved by forming its diastereomeric salt with an optically active organic acid, undergoing reduction of the ester moiety, isobutyrylation of the phenolic hydroxyl group, and fesoterodine and its (S) mirror image The isomer is produced. [Selection figure] None |
isCitedBy |
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2015520139-A |
priorityDate |
2009-10-29-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type |
http://data.epo.org/linked-data/def/patent/Publication |