http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2011064695-A

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filingDate 2010-11-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_54deb419faf8c690f3f20ca0d29d0a9c
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5a5dd0e9465f637896eecf088315eefc
publicationDate 2011-03-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2011064695-A
titleOfInvention Incontinence treatment
abstract The present invention provides a method for treating incontinence, an assay for screening compounds useful for the treatment of incontinence, and a method for producing a composition for treating urinary incontinence. A method for screening a compound useful for the treatment of stress urinary incontinence comprising the step of screening a compound for agonistic activity against 5-HT2C receptor and selecting a compound having an EC50 of less than 100 nM. Method. A process for providing a medicament for the treatment of stress urinary incontinence comprising the steps of: (a) testing the compound in a ligand binding assay for 5-HT2C receptor; (b) a compound having an IC50 of less than 100 nM. (C) formulating a compound having the same structure as the compound selected in step (b) or a pharmaceutically acceptable salt thereof together with a pharmaceutically acceptable carrier or excipient. process. [Selection figure] None
priorityDate 2003-04-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 463.