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filingDate 2010-10-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c49e16793652e8a84e7b09340967d061
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publicationDate 2011-03-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2011046731-A
titleOfInvention Water-soluble benzazepine compound and pharmaceutical composition
abstract An object of the present invention is to provide a novel benzoazepine compound having improved solubility of tolvaptan in water and suitable for use as an injection. The present invention provides a benzazepine compound represented by the following general formula (1) or a salt thereof. [Wherein, R represents a hydrogen atom, a hydroxy group having a protecting group, or the like. R 1 represents a hydrogen atom or a hydroxy protecting group. X represents an oxygen atom or a sulfur atom. ] [Selection figure] None
priorityDate 2005-12-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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