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filingDate 2010-08-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_28645ea80a4655523e294fc0a901d79a
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publicationDate 2011-02-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2011037857-A
titleOfInvention 6- (3-Chloro-2-fluorobenzyl) -1-[(2S) -1-hydroxy-3-methylbutan-2-yl] -7-methoxy-4-oxo for the treatment of retroviral infections Use of -1,4-dihydroquinoline-3-carboxylic acid or a salt thereof
abstract [PROBLEMS] To provide a therapeutic agent for retroviral infection, a therapeutic composition and a kit. A therapeutically effective amount of 6- (3-chloro-2-fluorobenzyl) -1-[(2S) -1-hydroxy-3-methylbutan-2-yl] -7-methoxy-4-oxo-1 , 4-Dihydroquinoline-3-carboxylic acid (hereinafter referred to as Compound I) or a pharmaceutically acceptable salt thereof. Furthermore, use of compound I or a salt thereof for an inhibitor of integrase activity. Compound I or salts thereof are also effective in inhibiting the replication of retroviruses that are resistant to at least one antiretroviral agent. Compound I or a salt thereof is administered alone or in combination with at least one antiretroviral agent other than Compound I or a salt thereof. Furthermore, manufacture of a kit containing Compound I or a salt thereof. [Selection figure] None
priorityDate 2006-02-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7JFM3
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP23989
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ95KP3
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID409863106
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0TKT1
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9R0J8
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP61756
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7CIZ3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP49676
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6LL68
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA7KGA5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP61757
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ07885
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP81800
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6395
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID403931
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP19593
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID114447
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8LKW0
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID411621736
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO14746
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135398508
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID12774
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2VHN8
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID450124
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5PXD0
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ27ID4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ865Y1
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID735311
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8A3N2
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8A4C3
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID464205
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID707329
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Total number of triples: 479.