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filingDate 2008-09-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2010-12-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2010540503-A
titleOfInvention Pyrazolo-pyrazine derivatives as G protein inhibitors
abstract The present invention relates to pyrazolo-pyrazine derivatives of general formula (I) Wherein Z, R 1 , R 2 , R 3 and R 4 groups represent variable groups, X is a sulfur atom or selenium atom, and n is an integer equal to 1 or 2. They are particularly important for the treatment of diseases involving heterotrimeric G proteins. The present invention also relates to pharmaceutical compositions comprising the product and their use to produce a drug.
priorityDate 2007-09-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID59474047
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ29450

Total number of triples: 312.