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filingDate 2008-09-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2010-12-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2010539945-A
titleOfInvention Antibodies against factor Xa inhibitors and methods of use thereof
abstract One of the main limitations of anticoagulant therapy is the risk of treatment-related bleeding and limited ability to rapidly reverse anticoagulant activity in the event of overdose or emergency surgical treatment . Therefore, a specific and effective antidote for all forms of anticoagulant therapy is highly desirable. The present invention relates to an antidote to an anticoagulant that targets factor Xa. An antidote is a factor Xa protein derivative that binds to and substantially neutralizes a factor Xa inhibitor but does not aggregate to form a prothrombinase complex. The derivatives described herein lack or have a reduced intrinsic clotting activity. Disclosed herein are methods for stopping or preventing bleeding in patients currently undergoing anticoagulation therapy with a factor Xa inhibitor.
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419559027
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID450133
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID20835957
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID10029
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID885074
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID856579
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP28842
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID13807
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID1551643
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID877794
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID411181230

Total number of triples: 644.