http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2010530862-A

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filingDate 2008-06-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2010-09-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2010530862-A
titleOfInvention Isoxazole-imidazole derivatives
abstract The present invention relates to isoxazole-imidazole derivatives having affinity and selectivity for GABA Aα5 receptor binding site, their production, pharmaceutical compositions containing them, and their use as pharmaceuticals. The active compounds of the present invention are useful as cognitive enhancers or in the treatment of cognitive disorders such as Alzheimer's disease. In particular, the invention provides an aryl-isoxazol-4-yl-imidazole derivative of formula I: wherein R 1 , R 2 and R 3 are as described in the specification.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2014502279-A
priorityDate 2007-06-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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