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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P43-00
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-428
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filingDate 2009-03-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b6bdcf6cda031a5581382299cca520bc
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_4e43ae7c07a59527beb7a622c0ee88f2
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publicationDate 2010-10-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2010229039-A
titleOfInvention Glyoxalase I inhibitor
abstract A glyoxalase I inhibitor having a novel skeleton different from a glutathione derivative and having high specificity for human glyoxalase I is provided. The present invention provides a glyoxalase I inhibitor and an anticancer agent represented by a predetermined general formula. The glyoxalase I inhibitor and anticancer agent of the present invention can inhibit the activity of human glyoxalase I with high specificity. For this reason, it can utilize effectively as a therapeutic agent of various diseases, such as an anticancer agent and an osteoporosis therapeutic agent. [Selection] Figure 10
priorityDate 2009-03-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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