http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2010090078-A

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assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_e13cf25eb1bef6199475314477618b46
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P9-10
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D498-04
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P3-06
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-553
filingDate 2008-10-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_d1db653734a3615490d9bd92ddf2a627
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8fd7c5bbbe578bc5f7ce0d3c77038df2
publicationDate 2010-04-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2010090078-A
titleOfInvention Tricyclic heteroaryl derivatives
abstract Hyperlipidemia such as hypercholesterolemia, hypertriglyceridemia, hypoHDLemia and the like for mammals including humans, exhibiting squalene synthase inhibitory activity, cholesterol synthesis inhibitory activity and low toxicity The provision of a compound useful as a pharmaceutical agent such as a prophylactic and / or therapeutic agent for arteriosclerosis. (1) [(4R, 6R) -8-chloro-6- (2-cyano-3-ethoxyphenyl) -1- (trifluoromethyl) -4H, 6H- [1,2,4] Triazolo [4,3-a] [4,1] benzoxazepin-4-yl] acetic acid (2) [(4R, 6R) -8-chloro-1- [chloro (difluoro) methyl] -6 -(2-cyano-3-methoxyphenyl) -4H, 6H- [1,2,4] triazolo [4,3-a] [4,1] benzoxazepin-4-yl] acetic acid, etc. Specific compound. [Selection figure] None
priorityDate 2008-10-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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