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filingDate 2007-05-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2009-10-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2009537570-A
titleOfInvention Unit dose formulation with inhalable solution of albuterol
abstract The present invention includes (a) preparing about 0.84 to about 0.90 wt% NaCl, (b) mixing the NaCl with about 80 wt% water to produce an aqueous solution, c) adding about 0.03 to about 0.25% by weight of albuterol free base to the solution of (b); (d) about 0.10 to about 1.3% by weight of HCl (1N) ( c) adding to the solution of (e), adding a sufficient amount of water to the solution of (e) (d) to make the total weight percent equal to 100, and (f) filtering the solution of (e). A unit dose formulation having a therapeutically effective amount of albuterol solution prepared by a process comprising sterilizing and dividing the solution of (g) (f) into unit doses of about 0.5 ml The molar ratio of albuterol free base: HCl is about 0. 5 to about 1.20, pH is about 3.0 to about 4.5, it has a therapeutically effective amount of albuterol and provides it has) suitable for inhalation therapy via nebulization.
priorityDate 2006-05-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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