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filingDate 2007-03-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2009-09-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2009531408-A
titleOfInvention Polymorphic form of olopatadine hydrochloride and process for producing olopatadine and its salts
abstract A method for producing olopatadine or a salt thereof by Wittig reaction of 11-oxo-6,11-dihydrodibenzo [b, e] oxepin-2-acetic acid and 3-dimethylaminopropyltriphenylphosphonium halide in the presence of a base, olopatadine or Method for increasing the (Z) / (E) ratio of a diastereomeric mixture containing the salt, 11-oxo-6,11-dihydrodibenzo [b, e] oxepin-2-acetic acid and 3-dimethylaminopropyltriphenyl Process for producing phosphonium bromide, and polymorph B of olopatadine hydrochloride. [Selection figure] None
priorityDate 2006-03-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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