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filingDate 2006-12-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2009-06-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2009522357-A
titleOfInvention Use of oripavine as a starting material for buprenorphine
abstract Here, a method of synthesis of norbuprenorphine and finally buprenorphine is provided, utilizing oripavine as a starting material. Conventional methods for producing buprenorphine utilize thebaine as a starting material and require an O-demethylation step, which is typically a low to medium yield conversion. Since oripavine molecules lack the O-3 methyl group, the use of oripavine as a starting material at this time does not require an O-demethylation step.
priorityDate 2006-01-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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