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filingDate 2006-12-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2009-05-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2009518404-A
titleOfInvention Androgen receptor modulator (N-3H-imidazo [4,5-B] pyridin-2-ylmethyl) -2-fluoro-4-methyl-3-oxo-4-aza-androst-1-en-17-beta Carboxamide polymorphs
abstract The compound of structural formula I is a tissue selective modulator of the androgen receptor (AR). These compounds can be used to strengthen reduced muscle tone, as well as osteoporosis, osteopenia, glucocorticoid-induced osteoporosis, periodontal disease, fractures, bone damage after bone reconstruction, myopathy, embrittlement, aging skin , Male hypogonadism, female postmenopausal symptoms, atherosclerosis, hypercholesterolemia, hyperlipidemia, obesity, irreproducible anemia and other hematopoietic disorders, inflammatory arthritis and joint repair, HIV Weakness, prostate cancer, benign prostatic hyperplasia (BPH), abdominal adiposity, metabolic syndrome, type II diabetes, cancer categorization, Alzheimer's disease, muscular dystrophy, cognitive decline, sexual dysfunction, sleep apnea, depression, premature ovary For the treatment of conditions caused by androgen deficiency, such as deficiencies and autoimmune diseases, or can be alleviated by androgen administration, alone or in combination with other active agents It is.
priorityDate 2005-12-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP80276
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01269
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID408184029
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9GMB3
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID54250
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID411746874
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID150311
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01268
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9GMB2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP09476
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP52212
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID395909
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID26585
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID105026
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID460178
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID373617
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426340844
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID397769
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCF1PKH2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ05700
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID406207
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1066
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01287
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID359834
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419554602
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP09477
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCF1PI70
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01286
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP09537
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID231
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCF1PM04
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419551077
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9W6J5
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419486648
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP09539
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID56637
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9W6R8
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6918123
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID444686
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419535788

Total number of triples: 1006.