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filingDate 2006-11-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2009-04-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2009515836-A
titleOfInvention [4- (6-halo-7-substituted-2,4-dioxo-1,4-dihydro-2H-quinazolin-3-yl) -phenyl] -5-chloro-thiophen-2-yl-sulfonylurea, and Related forms and methods
abstract The present invention provides novel sulfonylurea compounds of formula (I) and their pharmaceutically acceptable derivatives, polymorphic and amorphous forms. Various forms of these compounds are effective platelet ADP receptor inhibitors, can be used in various pharmaceutical compositions, and are particularly effective for the prevention and / or treatment of cardiovascular diseases, particularly those associated with thrombosis. Is. The present invention includes the steps of preparing such compounds and forms and administering a therapeutically effective amount of a compound of formula (I) or a pharmaceutically acceptable salt or form thereof, and thrombosis and thrombosis related in mammals Also provided are methods for preventing or treating a disease state.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-WO2014042176-A1
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2016026231-A
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http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2013544271-A
priorityDate 2005-11-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP80595
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID25095577
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID456459936
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0JND9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP23466
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6Z4P2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP96471
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ05766
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426299103
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419525604
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419860824
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO93295
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ99396
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP00749
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID424318167
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7299

Total number of triples: 327.