http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2009504627-A
Outgoing Links
| Predicate | Object |
|---|---|
| classificationCPCAdditional | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/Y02P20-55 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D487-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P43-00 |
| classificationIPCAdditional | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07B61-00 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P43-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-407 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D487-04 |
| filingDate | 2006-08-10-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 2009-02-05-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | JP-2009504627-A |
| titleOfInvention | Preparation of diazapentane via epoxy reaction of dihydropyrrole |
| abstract | The present invention relates to a method for preparing a compound of the following formula (I), or a pharmaceutically acceptable salt thereof: Here in the formula, R 1 is an Pg 1 or P 1 '; P 1 ′ is CO-hydrocarbyl (Hydrocarbyl); P 2 is CH 2 , O or N—Pg 2 ; and Pg 1 and Pg 2 are each independently a nitrogen protecting group; The method comprises the following steps: (I) reacting dioxirane with a compound of formula II to form an epoxide of formula III (i); Here in the formula, X, CN, is selected from CH 2 N 3, CH 2 NH -Pg 2, ONH-Pg 2, NHNH-Pg 2, and N (Pg 2) NH-Pg 2; (Ii) converting the compound of formula III to the compound of formula I (ii) About. |
| priorityDate | 2005-08-10-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 279.