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filingDate 2006-06-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2009-01-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2009500338-A
titleOfInvention Compound
abstract The present invention relates to a novel indole carboxamide derivative. In particular, the present invention provides compounds of formula (I): [Wherein R1, R2, R3, U and V are defined below] And a pharmaceutically acceptable salt thereof. The compounds of the invention are inhibitors of IKK2 and are useful in the treatment of disorders associated with inappropriate IKK2 (also known as IKKβ) activity such as rheumatoid arthritis, asthma, and COPD (chronic obstructive pulmonary disease). sell. Accordingly, the present invention further relates to pharmaceutical compositions comprising the compounds of the present invention. The invention further relates to a method of inhibiting IKK2 activity and a method of treating disorders associated with the use of a compound of the invention or a pharmaceutical composition comprising the invention.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2021001212-A
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2017531679-A
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http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2019123740-A
priorityDate 2005-06-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421504429
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66723272
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP17928
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66723249
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421504427
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415759023
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16036915
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8R8N1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO49564
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID452521482
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421504433
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID281073
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426129961
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66723274
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8R5N8
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16036914
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66723251
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421504431
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID420461051
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID454435913
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66723277
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66723250
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421504436
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10129899
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16036916
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP18061
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10396794
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66723221
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421504434
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450686317
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426027762
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID447554
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66723220
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421504440
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5126
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1956
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6999786
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421504438
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419490211
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID452557052
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415905233
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID422059129
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3JW78
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID410535579
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66723280
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66723345
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID413144997
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID448769946
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6999788
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426218560
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3K1W9
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66723282
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421145748
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5I6E3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3B2F5
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419519592
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7150
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66723229
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6PUD2
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66723228
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID153678241
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID448716735
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID13003
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66723231
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16037739
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3BQW1
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID448719745
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415763186
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16037741
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID465664045
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID151411
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID448719255
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66723259
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID452431749
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP41683
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16037740
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419593536
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID454354489
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66723235
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID300809
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16037743
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID448720737
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66723261
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6R2X3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP41693
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3E9X6
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP41687
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID465687963
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66723263
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA8I1Q0
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12246
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8P709
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421586839
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421504086

Total number of triples: 2921.