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publicationDate 2009-07-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2009155342-A
titleOfInvention Cytotoxins, prodrugs, linkers and useful stabilizers
abstract Disclosed is a compound exhibiting high action specificity and low toxicity as compared with known compounds having a similar structure and improved blood stability. A linker arm is provided that liberates an active drug moiety from a prodrug derivative that is cleaved enzymatically or reductively in vivo to include a linker arm. The linker arm further includes conjugates between cytotoxins and linker arms, conjugates between cytotoxins and targeting agents such as antibodies or peptides. [Selection figure] None
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Total number of triples: 447.