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filingDate 2006-05-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2008-11-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2008540618-A
titleOfInvention Peptidomimetics selective for somatostatin receptor subtype 1 and / or 4
abstract The present invention defines Formula (I) {A, D, E, J, Q, R1, R2, R3, p, and j in the formula as disclosed. }, A (hetero) arylsulfonylamino-based peptidomimetic, or a pharmaceutically acceptable salt or ester thereof. Compounds represented by formula (I) have a high affinity and selectivity for somatostatin receptor subtypes sst 1 and / or sst 4, agonists or antagonists of sst 1 and / or sst 4 is useful It can be used to treat or diagnose a disease or condition that has been suggested.
priorityDate 2005-05-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 731.