http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2008532996-A
Outgoing Links
| Predicate | Object |
|---|---|
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D513-06 |
| classificationIPCAdditional | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-542 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07B61-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D513-06 |
| filingDate | 2005-06-23-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 2008-08-21-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | JP-2008532996-A |
| titleOfInvention | Synthetic methods of substituted benzothiazinoindoles |
| abstract | General formula (I) [wherein R 1 , R 2 and R 4 are independently hydrogen, chlorine, fluorine, amino, nitro, cyano, CHO, (C 1 -C 3 ) alkyl, perfluoro (C 1 -C 3) alkyl, (C 1 ~C 3) alkoxy, aryl, aralkyl, aralkoxy, (C 5 ~C 7) heterocyclyl, (C 5 ~C 7) heterocyclylalkyl, (C 5 ~C 7) heterocyclyloxy , Acyl, acetyl, alkylamino, aminoalkyl, amide, hydroxyalkyl, carboxylic acid groups and derivatives thereof, R 3 is hydrogen, (C 1 -C 3 ) alkyl, aryl, and carboxylic acid groups and derivatives thereof A method for the synthesis of substituted benzothiazinoindoles is selected. The method involves the cyclization of a compound of general formula (II) (ie substituted 1-benzenesulfonyl-7-bromo-1H-indole) using an appropriate catalyst and solvent. |
| priorityDate | 2005-03-08-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 100.