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filingDate 2006-02-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2008-08-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2008531689-A
titleOfInvention 2- [Isoquinoline-3-carbonyl) amino] -propionic acid derivatives as inhibitors of factor XI and factor IX for the treatment of thrombosis
abstract The present invention relates to formula (X) [Chemical 1] Aryl and heteroaryl compounds of the invention are provided. The compounds of the present invention are useful as antagonists or factor IX and / or partial antagonists of factor XI and can be used to inhibit the intrinsic pathway of blood clotting. In the formula (X), R 102 represents —C (O) OH, —C (O) OCH 3 , —C (O) Ot-butyl, —C (O) NH—OCH 2 -phenyl, C ( R 101 , R 103 , R 104 and Y are defined herein, selected from the group consisting of O) NHOH and —C (O) NHSO 2 CH 3 .
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2013501074-A
priorityDate 2005-03-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 563.