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filingDate 2005-10-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2008-06-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2008518925-A
titleOfInvention Liposome preparation process
abstract The present invention provides a process for producing a liposomal formulation comprising a water-insoluble or hydrophobic active principle. In one embodiment of the method of the present invention, at least one active principle and lipid fraction are dissolved in an organic solvent. This solution is then subjected to reduced pressure (vacuum) in an inertly packaged or not container to remove the organic solvent, resulting in the formation of a puff cake containing the active ingredient and lipid fraction. This puff cake is then mixed with the aqueous solution under controlled conditions suitable to form a bulk liposome formulation. Since the effective main component is contained in the lipid bilayer, the removal of the aqueous solution is optional. [Selection] Figure 1
priorityDate 2004-10-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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